Found 735 of ec50 for Vasopressin receptor
having polymerids = 325,326,4332,49001080,49001083 and
complexids = 50013946
having polymerids = 325,326,4332,49001080,49001083 and
complexids = 50013946
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 0.00400nMAssay Description:Agonist activity at recombinant human V1a receptor expressed in HEK293 cells assessed as increase in intracellular calcium level measured at 3 secs i...More data for this Ligand-Target Pair
Affinity DataEC50: 0.0200nMAssay Description:Agonist activity at recombinant rat V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ge...More data for this Ligand-Target Pair
Affinity DataEC50: 0.0300nMAssay Description:Agonist activity at recombinant rat V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ge...More data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 0.0340nMAssay Description:Agonist activity at human V1b receptor expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
Affinity DataEC50: 0.0500nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
Affinity DataEC50: 0.0500nMAssay Description:Agonist activity at human vasopressin V2 expressed in HEK293 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0500nMAssay Description:Agonist activity at recombinant rat V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ge...More data for this Ligand-Target Pair
Affinity DataEC50: 0.0700nMAssay Description:Agonist activity at recombinant rat vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0700nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
Affinity DataEC50: 0.0800nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
Affinity DataEC50: 0.0800nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
Affinity DataEC50: 0.100nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
Affinity DataEC50: 0.100nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
Affinity DataEC50: 0.100nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
Affinity DataEC50: 0.100nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
Affinity DataEC50: 0.100nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
Affinity DataEC50: 0.105nMAssay Description:Agonist activity at recombinant rat vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.110nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
Affinity DataEC50: 0.120nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 0.120nMAssay Description:Agonist activity at human V1a receptor expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
Affinity DataEC50: 0.123nMAssay Description:Agonist activity at recombinant rat vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 0.126nMAssay Description:Compound was evaluated for in vitro potency against angiotensin II receptor, type 1 in isolated rabbit aorta; value ranges from 8.27-8.70More data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 0.126nMAssay Description:Compound was evaluated for in vitro potency against AT1 receptor in isolated rabbit aorta; value ranges from 7.91-7.97More data for this Ligand-Target Pair
Affinity DataEC50: 0.126nMAssay Description:Agonist activity at recombinant rat vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.140nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 0.140nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 0.155nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 0.158nMAssay Description:Compound was evaluated for in vitro potency against angiotensin II receptor, type 1 in isolated rabbit aortaMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 0.158nMAssay Description:In vitro for histamine H1 receptor antagonist activity against histamine-induced contractions on isolated guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: 0.162nMAssay Description:Agonist activity at recombinant rat vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.170nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 0.170nMAssay Description:Agonist activity at human V1b receptor expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 0.180nMAssay Description:Agonist activity at human V1A receptor expressed in HEK293 cells assessed as intracellular calcium level measured at 3 secs interval for 5 mins by fu...More data for this Ligand-Target Pair
Affinity DataEC50: 0.190nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 0.190nMAssay Description:Agonist activity at recombinant human V1a receptor expressed in HEK293 cells assessed as increase in intracellular calcium level measured at 3 secs i...More data for this Ligand-Target Pair
Affinity DataEC50: 0.190nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
Affinity DataEC50: 0.190nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
Affinity DataEC50: 0.200nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
Affinity DataEC50: 0.200nMAssay Description:Agonist activity at human vasopressin V2 expressed in HEK293 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.200nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
Affinity DataEC50: 0.210nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
Affinity DataEC50: 0.210nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 0.210nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.220nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
Affinity DataEC50: 0.220nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
Affinity DataEC50: 0.220nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
Affinity DataEC50: 0.230nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
Affinity DataEC50: 0.230nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 0.234nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Tohoku University And Department Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataEC50: 0.240nMAssay Description:Agonist activity at human vasopressin V1a expressed in HEK293 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair